| Reaction Details |
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 | Report a problem with these data |
| Target | D(1A) dopamine receptor |
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| Ligand | BDBM50289539 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_58299 |
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| IC50 | >10000±n/a nM |
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| Citation |  Mantegani, S; Brambilla, E; Cremonesi, P; Caccia, C; Fornaretto, MG; Carfagna, N; Colombo, M; McArthur, RA; Varasi, M (E) and (Z)-3-Styrylpiperidines as sigma ligands Bioorg Med Chem Lett7:1525-1530 (1997) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(1A) dopamine receptor |
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| Name: | D(1A) dopamine receptor |
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| Synonyms: | DOPAMINE D1 | DRD1_RAT | Dopamine D1 high | Dopamine D1 low | Dopamine receptor | Dopamine receptor D1 | Dopamine1-like | Drd1 | Drd1a |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 49429.75 |
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| Organism: | RAT |
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| Description: | P18901 |
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| Residue: | 446 |
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| Sequence: | MAPNTSTMDEAGLPAERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNF
FVISLAVSDLLVAVLVMPWKAVAEIAGFWPLGPFCNIWVAFDIMCSTASILNLCVISVDR
YWAISSPFQYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTWPLDGNFTSLED
TEDDNCDTRLSRTYAISSSLISFYIPVAIMIVTYTSIYRIAQKQIRRISALERAAVHAKN
CQTTAGNGNPVECAQSESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFISNCMVPFCGS
EETQPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFQKAFSTLLGCYRLCPTTNNAIET
VSINNNGAVVFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKKEEAGGIAKPLEKLSPAL
SVILDYDTDVSLEKIQPVTHSGQHST
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| BDBM50289539 |
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| n/a |
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| Name | BDBM50289539 |
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| Synonyms: | 1-Cyclohexyl-3-((Z)-styryl)-piperidine | CHEMBL39806 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H27N |
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| Mol. Mass. | 269.4244 |
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| SMILES | C1CCC(CC1)N1CCCC(C1)\C=C/c1ccccc1 |
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| Structure | 
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