Reaction Details |
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Target | Sigma non-opioid intracellular receptor 1 |
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Ligand | BDBM50289541 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEBML_201293 |
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IC50 | 4±n/a nM |
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Citation | Mantegani, S; Brambilla, E; Cremonesi, P; Caccia, C; Fornaretto, MG; Carfagna, N; Colombo, M; McArthur, RA; Varasi, M (E) and (Z)-3-Styrylpiperidines as sigma ligands Bioorg Med Chem Lett7:1525-1530 (1997) Article |
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More Info.: | Get all data from this article, Assay Method |
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Sigma non-opioid intracellular receptor 1 |
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Name: | Sigma non-opioid intracellular receptor 1 |
Synonyms: | Opioid receptor | Oprs1 | SGMR1_RAT | Sigma | Sigma non-opioid intracellular receptor 1 | Sigma opioid receptor | Sigma-1 | Sigmar1 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 25266.54 |
Organism: | RAT |
Description: | Q9R0C9 |
Residue: | 223 |
Sequence: | MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
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BDBM50289541 |
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n/a |
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Name | BDBM50289541 |
Synonyms: | 1-(3-Phenyl-propyl)-3-((E)-styryl)-piperidine | CHEMBL37661 |
Type | Small organic molecule |
Emp. Form. | C22H27N |
Mol. Mass. | 305.4565 |
SMILES | C(CN1CCCC(C1)\C=C\c1ccccc1)Cc1ccccc1 |
Structure |
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