| Reaction Details |
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 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 5 |
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| Ligand | BDBM50148348 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_608576 (CHEMBL1065841) |
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| EC50 | 12±n/a nM |
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| Citation |  Lu, Y; Wang, Z; Li, CM; Chen, J; Dalton, JT; Li, W; Miller, DD Synthesis, in vitro structure-activity relationship, and in vivo studies of 2-arylthiazolidine-4-carboxylic acid amides as anticancer agents. Bioorg Med Chem18:477-95 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Lysophosphatidic acid receptor 5 |
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| Name: | Lysophosphatidic acid receptor 5 |
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| Synonyms: | GPR92 | GPR93 | LPAR5 | LPAR5_HUMAN | Lysophosphatidic acid receptor 5 | Lysophosphatidic acid receptor 5 (LPA5) |
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| Type: | Enzyme |
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| Mol. Mass.: | 41372.36 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q9H1C0 |
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| Residue: | 372 |
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| Sequence: | MLANSSSTNSSVLPCPDYRPTHRLHLVVYSLVLAAGLPLNALALWVFLRALRVHSVVSVY
MCNLAASDLLFTLSLPVRLSYYALHHWPFPDLLCQTTGAIFQMNMYGSCIFLMLINVDRY
AAIVHPLRLRHLRRPRVARLLCLGVWALILVFAVPAARVHRPSRCRYRDLEVRLCFESFS
DELWKGRLLPLVLLAEALGFLLPLAAVVYSSGRVFWTLARPDATQSQRRRKTVRLLLANL
VIFLLCFVPYNSTLAVYGLLRSKLVAASVPARDRVRGVLMVMVLLAGANCVLDPLVYYFS
AEGFRNTLRGLGTPHRARTSATNGTRAALAQSERSAVTTDATRPDAASQGLLRPSDSHSL
SSFTQCPQDSAL
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| BDBM50148348 |
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| n/a |
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| Name | BDBM50148348 |
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| Synonyms: | (R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-propyl ester | 1-oleoyl lysophosphatidic acid | CHEMBL117021 | lysophosphatidic acid |
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| Type | Small organic molecule |
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| Emp. Form. | C21H41O7P |
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| Mol. Mass. | 436.5198 |
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| SMILES | CCCCCCCC\C=C/CCCCCCCC(=O)OC[C@@H](O)COP(O)(O)=O |
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| Structure | 
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