| Reaction Details |
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 | Report a problem with these data |
| Target | Glucagon-like peptide 1 receptor |
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| Ligand | BDBM50314040 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_626670 (CHEMBL1108872) |
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| IC50 | 10.1±n/a nM |
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| Citation |  Son, S; Chae, SY; Kim, CW; Choi, YG; Jung, SY; Lee, S; Lee, KC Preparation and structural, biochemical, and pharmaceutical characterizations of bile acid-modified long-acting exendin-4 derivatives. J Med Chem52:6889-96 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Glucagon-like peptide 1 receptor |
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| Name: | Glucagon-like peptide 1 receptor |
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| Synonyms: | GLP1R_RAT | Glp1r | Glpr |
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| Type: | PROTEIN |
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| Mol. Mass.: | 52889.73 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_855307 |
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| Residue: | 463 |
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| Sequence: | MAVTPSLLRLALLLLGAVGRAGPRPQGATVSLSETVQKWREYRHQCQRFLTEAPLLATGL
FCNRTFDDYACWPDGPPGSFVNVSCPWYLPWASSVLQGHVYRFCTAEGIWLHKDNSSLPW
RDLSECEESKQGERNSPEEQLLSLYIIYTVGYALSFSALVIASAILVSFRHLHCTRNYIH
LNLFASFILRALSVFIKDAALKWMYSTAAQQHQWDGLLSYQDSLGCRLVFLLMQYCVAAN
YYWLLVEGVYLYTLLAFSVFSEQRIFKLYLSIGWGVPLLFVIPWGIVKYLYEDEGCWTRN
SNMNYWLIIRLPILFAIGVNFLVFIRVICIVIAKLKANLMCKTDIKCRLAKSTLTLIPLL
GTHEVIFAFVMDEHARGTLRFVKLFTELSFTSFQGFMVAVLYCFVNNEVQMEFRKSWERW
RLERLNIQRDSSMKPLKCPTSSVSSGATVGSSVYAATCQNSCS
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| BDBM50314040 |
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| n/a |
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| Name | BDBM50314040 |
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| Synonyms: | CHEMBL1092707 |
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| Type | Small organic molecule |
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| Emp. Form. | C232H357N49O67S |
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| Mol. Mass. | 4936.67 |
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| SMILES | n/a |
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| Structure | 
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