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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Glutamate receptor 3 | ||
| Ligand | BDBM50316375 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEMBL_628117 (CHEMBL1108128) | ||
| EC50 | 1660±n/a nM | ||
| Citation |  Fleming, JJ; England, PM Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands. Bioorg Med Chem18:1381-7 (2010) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Glutamate receptor 3 | |||
| Name: | Glutamate receptor 3 | ||
| Synonyms: | AMPA-selective glutamate receptor 3 | GLUR3 | GLURC | GRIA3 | GRIA3_HUMAN | GluR-3 | GluR-C | GluR-K3 | Glutamate receptor 3 | Glutamate receptor ionotropic AMPA | Glutamate receptor ionotropic, AMPA 3 | ||
| Type: | PROTEIN | ||
| Mol. Mass.: | 101172.14 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | ChEMBL_468627 | ||
| Residue: | 894 | ||
| Sequence: |
| ||
| BDBM50316375 | |||
| n/a | |||
| Name | BDBM50316375 | ||
| Synonyms: | CHEMBL1097939 | LY-404187 | N-[2-(4'-cyanobiphenyl-4-yl)propyl]propane-2-sulfonamide | ||
| Type | Small organic molecule | ||
| Emp. Form. | C19H28N2O2S | ||
| Mol. Mass. | 348.503 | ||
| SMILES | CC(C)S(=O)(=O)NCC(C)C1CCC(CC1)c1ccc(cc1)C#N |(35.08,-18.3,;35.1,-19.84,;36.44,-20.59,;33.78,-20.62,;32.99,-21.94,;34.53,-21.94,;32.44,-19.86,;31.11,-20.63,;29.77,-19.86,;29.77,-18.32,;28.44,-20.63,;28.44,-22.17,;27.12,-22.94,;25.78,-22.17,;25.77,-20.64,;27.1,-19.86,;24.45,-22.95,;23.11,-22.18,;21.79,-22.95,;21.79,-24.5,;23.12,-25.27,;24.46,-24.5,;20.45,-25.27,;19.11,-26.03,)| | ||
| Structure | 
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