| Reaction Details |
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 | Report a problem with these data |
| Target | P2Y purinoceptor 11 |
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| Ligand | BDBM50347445 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_755242 (CHEMBL1806221) |
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| EC50 | 13000±n/a nM |
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| Citation |  Eliahu, S; Lecka, J; Reiser, G; Haas, M; Bigonnesse, F; Lévesque, SA; Pelletier, J; Sévigny, J; Fischer, B Diadenosine 5',5''-(boranated)polyphosphonate analogues as selective nucleotide pyrophosphatase/phosphodiesterase inhibitors. J Med Chem53:8485-97 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| P2Y purinoceptor 11 |
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| Name: | P2Y purinoceptor 11 |
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| Synonyms: | P2RY11 | P2Y purinoceptor 11 | P2Y11 | P2Y11_HUMAN | Purinergic receptor P2Y11 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 40366.02 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1362532 |
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| Residue: | 374 |
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| Sequence: | MAANVSGAKSCPANFLAAADDKLSGFQGDFLWPILVVEFLVAVASNGLALYRFSIRKQRP
WHPAVVFSVQLAVSDLLCALTLPPLAAYLYPPKHWRYGEAACRLERFLFTCNLLGSVIFI
TCISLNRYLGIVHPFFARSHLRPKHAWAVSAAGWVLAALLAMPTLSFSHLKRPQQGAGNC
SVARPEACIKCLGTADHGLAAYRAYSLVLAGLGCGLPLLLTLAAYGALGRAVLRSPGMTV
AEKLRVAALVASGVALYASSYVPYHIMRVLNVDARRRWSTRCPSFADIAQATAALELGPY
VGYQVMRGLMPLAFCVHPLLYMAAVPSLGCCCRHCPGYRDSWNPEDAKSTGQALPLNATA
APKPSEPQSRELSQ
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| BDBM50347445 |
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| n/a |
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| Name | BDBM50347445 |
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| Synonyms: | CHEMBL1802094 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H31BN10O19P5 |
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| Mol. Mass. | 905.22 |
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| SMILES | [BH3-]P(=O)(OP([O-])(=O)CP([O-])(=O)OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)OP([O-])(=O)CP([O-])(=O)OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12 |r| |
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| Structure | 
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