| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide Y receptor type 5 |
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| Ligand | BDBM50355854 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_775144 (CHEMBL1912449) |
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| Ki | 1.8±n/a nM |
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| Citation |  Packiarajan, M; Coate, H; Desai, M; Jimenez, HN; Reinhard, EJ; Jubian, VJ; Marzabadi, MR; Chandrasena, G; Wolinski, TC; Walker, MW; Andersen, K 5-(2'-Pyridyl)-2-aminothiazoles: alkyl amino sulfonamides and sulfamides as potent NPY(5) antagonists. Bioorg Med Chem Lett21:6500-4 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Neuropeptide Y receptor type 5 |
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| Name: | Neuropeptide Y receptor type 5 |
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| Synonyms: | NPY-Y5 | NPY-Y5 receptor | NPY5-R | NPY5R | NPY5R_HUMAN | NPYR5 | NPYY5 | Neuropeptide Y receptor type 5 | Neuropeptide Y receptor type 5 ( NPY Y5) | Y5 receptor |
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| Type: | Enzyme |
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| Mol. Mass.: | 50746.64 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q15761 |
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| Residue: | 445 |
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| Sequence: | MDLELDEYYNKTLATENNTAATRNSDFPVWDDYKSSVDDLQYFLIGLYTFVSLLGFMGNL
LILMALMKKRNQKTTVNFLIGNLAFSDILVVLFCSPFTLTSVLLDQWMFGKVMCHIMPFL
QCVSVLVSTLILISIAIVRYHMIKHPISNNLTANHGYFLIATVWTLGFAICSPLPVFHSL
VELQETFGSALLSSRYLCVESWPSDSYRIAFTISLLLVQYILPLVCLTVSHTSVCRSISC
GLSNKENRLEENEMINLTLHPSKKSGPQVKLSGSHKWSYSFIKKHRRRYSKKTACVLPAP
ERPSQENHSRILPENFGSVRSQLSSSSKFIPGVPTCFEIKPEENSDVHELRVKRSVTRIK
KRSRSVFYRLTILILVFAVSWMPLHLFHVVTDFNDNLISNRHFKLVYCICHLLGMMSCCL
NPILYGFLNNGIKADLVSLIHCLHM
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| BDBM50355854 |
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| n/a |
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| Name | BDBM50355854 |
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| Synonyms: | CHEMBL1909727 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H27N5O2S2 |
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| Mol. Mass. | 397.559 |
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| SMILES | CCN(CC)S(=O)(=O)NCCCCCNc1nc(cs1)-c1ccccn1 |
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| Structure | 
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