| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50016086 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_145304 |
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| Ki | 31±n/a nM |
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| Citation |  Archer, S; Seyed-Mozaffari, A; Ward, S; Kosterlitz, HW; Paterson, SJ; McKnight, AT; Corbett, AD 10-Ketonaltrexone and 10-ketooxymorphone. J Med Chem28:974-6 (1985) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50016086 |
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| n/a |
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| Name | BDBM50016086 |
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| Synonyms: | 4-cyclopropylmethyl-10,17-dihydroxy-(13R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-triene-6,14-dione(Ketonaltrexone) | CHEMBL366520 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H21NO5 |
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| Mol. Mass. | 355.3844 |
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| SMILES | Oc1ccc2c3c1O[C@H]1C(=O)CC[C@@]4(O)C(N(CC5CC5)CCC314)C2=O |TLB:14:13:5.24.4:16.22.21,6:5:13:16.22.21,THB:25:24:13:16.22.21| |
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| Structure | 
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