Ki Summary BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetSerine protease 1
LigandBDBM50100969
Substrate/Competitorn/a
Meas. Tech.ChEBML_212532
Ki 5888437±n/a nM
Citation Yang, HHenkin, JKim, KHGreer, J Selective inhibition of urokinase by substituted phenylguanidines: quantitative structure-activity relationship analyses. J Med Chem33:2956-61 (1990) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Serine protease 1
Name:Serine protease 1
Synonyms:Beta-Trypsin | Cationic trypsin | PRSS1 | TRP1 | TRY1 | TRY1_BOVIN | TRYP1 | Trypsin | Trypsin I
Type:Enzyme
Mol. Mass.:25790.52
Organism:Bos taurus (bovine)
Description:P00760
Residue:246
Sequence:
MKTFIFLALLGAAVAFPVDDDDKIVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVS
AAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLN
SRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQIT
SNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIK
QTIASN
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50100969
n/a
NameBDBM50100969
Synonyms:1N-amino(immino)methyl-4-methoxyaniline | CHEMBL297076 | N-(4-Methoxy-phenyl)-guanidine | N-(4-methoxyphenyl)guanidine
TypeSmall organic molecule
Emp. Form.C8H11N3O
Mol. Mass.165.1924
SMILES[#6]-[#8]-c1ccc(cc1)\[#7]=[#6](\[#7])-[#7]
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: