| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50006946 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_145287 (CHEMBL752956) |
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| Ki | >1000±n/a nM |
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| Citation |  Portoghese, PS An approach to the design of receptor-type-selective non-peptide antagonists of peptidergic receptors: delta opioid antagonists. J Med Chem34:1757-62 (1991) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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|
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| BDBM50006946 |
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| n/a |
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| Name | BDBM50006946 |
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| Synonyms: | 2-[2-(2-{2-[2-Diallylamino-3-(4-hydroxy-phenyl)-propionylamino]-2-methyl-propionylamino}-2-methyl-propionylamino)-3-phenyl-propionylamino]-4-methyl-pentanoic acid | CHEMBL47545 | ICI-174864 |
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| Type | Small organic molecule |
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| Emp. Form. | C38H53N5O7 |
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| Mol. Mass. | 691.8567 |
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| SMILES | CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)C(C)(C)NC(=O)C(C)(C)NC(=O)[C@H](Cc1ccc(O)cc1)N(CC=C)CC=C)C(O)=O |
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| Structure | 
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