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TargetS-methyl-5'-thioadenosine phosphorylase
LigandBDBM50368300
Substrate/Competitorn/a
Meas. Tech.ChEBML_103126
Ki 26000±n/a nM
Citation Sufrin, JRSpiess, AJKramer, DLLibby, PRMiller, JTBernacki, RJLee, YHBorchardt, RTPorter, CW Targeting 5'-deoxy-5'-(methylthio)adenosine phosphorylase by 5'-haloalkyl analogues of 5'-deoxy-5'-(methylthio)adenosine. J Med Chem34:2600-6 (1991) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
S-methyl-5'-thioadenosine phosphorylase
Name:S-methyl-5'-thioadenosine phosphorylase
Synonyms:MTAP_MOUSE | Mtap | S-methyl-5-thioadenosine phosphorylase
Type:PROTEIN
Mol. Mass.:31064.59
Organism:Mus musculus
Description:ChEMBL_12784
Residue:283
Sequence:
MASGSACTAVKIGIIGGTGLDDPEILEGRTEKYVDTPFGKPSDALILGKIKNVDCVLLAR
HGRQHTIMPSKVNYQANIWALKEEGCTHVIVTTACGSLREEIQPGDMVIIDQFIDRTSLR
PQTFYDGSHCSARGVCHIPMAEPFCPKTREVLIETAKKLGLRCHSKGTIVTIEGPRFSSR
AESLIFRTWGADVVNMTTVPEVVLAKEAGICYASIAMATDYDCWKEHEEAVSVDGVLKTM
KENANKAKSLLLTTIPQIGSMEWSETLRNLKNMAQFSVLPPRH
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  Blast E-value cutoff:
BDBM50368300
n/a
NameBDBM50368300
Synonyms:CHEMBL608307
TypeSmall organic molecule
Emp. Form.C12H17N5O4S
Mol. Mass.327.359
SMILESNc1ncnc2n(cnc12)C1O[C@H](CSCCO)[C@@H](O)[C@H]1O |r|
Structure
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