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TargetLeukotriene B4 receptor 1
LigandBDBM50042148
Substrate/Competitorn/a
Meas. Tech.ChEBML_99839
Ki 60±n/a nM
Citation Kingsbury, WDPendrak, ILeber, JDBoehm, JCMallet, BSarau, HMFoley, JJSchmidt, DBDaines, RA Synthesis of structural analogs of leukotriene B4 and their receptor binding activity. J Med Chem36:3308-20 (1993) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Leukotriene B4 receptor 1
Name:Leukotriene B4 receptor 1
Synonyms:BLT | BLT1 | BLTR | CMKRL1 | Chemoattractant receptor-like 1 | G-protein coupled receptor 16 | GPR16 | LT4R1_HUMAN | LTB4-R 1 | LTB4R | Leukotriene B4 R1 | Leukotriene B4 receptor | Leukotriene B4 receptor 1 | P2RY7 | P2Y purinoceptor 7 | P2Y7
Type:Enzyme Catalytic Domain
Mol. Mass.:37582.68
Organism:Homo sapiens (Human)
Description:Q15722
Residue:352
Sequence:
MNTTSSAAPPSLGVEFISLLAIILLSVALAVGLPGNSFVVWSILKRMQKRSVTALMVLNL
ALADLAVLLTAPFFLHFLAQGTWSFGLAGCRLCHYVCGVSMYASVLLITAMSLDRSLAVA
RPFVSQKLRTKAMARRVLAGIWVLSFLLATPVLAYRTVVPWKTNMSLCFPRYPSEGHRAF
HLIFEAVTGFLLPFLAVVASYSDIGRRLQARRFRRSRRTGRLVVLIILTFAAFWLPYHVV
NLAEAGRALAGQAAGLGLVGKRLSLARNVLIALAFLSSSVNPVLYACAGGGLLRSAGVGF
VAKLLEGTGSEASSTRRGGSLGQTARSGPAALEPGPSESLTASSPLKLNELN
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  Blast E-value cutoff:
BDBM50042148
n/a
NameBDBM50042148
Synonyms:CHEMBL111811 | Lithium; 3-{1-hydroxy-2-[6-(3-hydroxy-undecyl)-pyridin-2-yl]-ethyl}-benzoate
TypeSmall organic molecule
Emp. Form.C25H34NO4
Mol. Mass.412.5423
SMILESCCCCCCCCC(O)CCc1cccc(CC(O)c2cccc(c2)C([O-])=O)n1
Structure
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