| Reaction Details |
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 | Report a problem with these data |
| Target | 3',5'-cyclic-AMP phosphodiesterase |
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| Ligand | BDBM50020874 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_155847 (CHEMBL766943) |
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| IC50 | 37200±n/a nM |
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| Citation |  Takase, Y; Saeki, T; Fujimoto, M; Saito, I Cyclic GMP phosphodiesterase inhibitors. 1. The discovery of a novel potent inhibitor, 4-((3,4-(methylenedioxy)benzyl)amino)-6,7,8-trimethoxyquinazoline. J Med Chem36:3765-70 (1994) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| 3',5'-cyclic-AMP phosphodiesterase |
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| Name: | 3',5'-cyclic-AMP phosphodiesterase |
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| Synonyms: | Phosphodiesterase 4A |
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| Type: | PROTEIN |
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| Mol. Mass.: | 13615.65 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_155848 |
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| Residue: | 118 |
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| Sequence: | PWLVGWWDQFKRMLNRELTHLSEMSRSGNQVSEYISTTFLDKQNEVDIPSPTMKDHEKQQ
APRQRPSQQPPPPGPQFQPMSQITGVKKLMHSSSLNEDSSIPRFGVKTDQEELLAQEL
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|
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| BDBM50020874 |
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| n/a |
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| Name | BDBM50020874 |
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| Synonyms: | (3-Chloro-phenyl)-(4-phenyl-phthalazin-1-yl)-amine | CHEMBL332898 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H14ClN3 |
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| Mol. Mass. | 331.798 |
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| SMILES | Clc1cccc(Nc2nnc(-c3ccccc3)c3ccccc23)c1 |
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| Structure | 
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