| Reaction Details |
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 | Report a problem with these data |
| Target | Melanocortin receptor 3 |
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| Ligand | BDBM50058956 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_106014 (CHEMBL716370) |
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| IC50 | >10000±n/a nM |
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| Citation |  Haskell-Luevano, C; Hendrata, S; North, C; Sawyer, TK; Hadley, ME; Hruby, VJ; Dickinson, C; Gantz, I Discovery of prototype peptidomimetic agonists at the human melanocortin receptors MC1R and MC4R. J Med Chem40:2133-9 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Melanocortin receptor 3 |
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| Name: | Melanocortin receptor 3 |
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| Synonyms: | MC3-R | MC3R | MC3R_HUMAN | Melanocortin MC3 | Melanocortin receptor (M3 and M4) |
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| Type: | Enzyme |
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| Mol. Mass.: | 36044.86 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P41968 |
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| Residue: | 323 |
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| Sequence: | MNASCCLPSVQPTLPNGSEHLQAPFFSNQSSSAFCEQVFIKPEVFLSLGIVSLLENILVI
LAVVRNGNLHSPMYFFLCSLAVADMLVSVSNALETIMIAIVHSDYLTFEDQFIQHMDNIF
DSMICISLVASICNLLAIAVDRYVTIFYALRYHSIMTVRKALTLIVAIWVCCGVCGVVFI
VYSESKMVIVCLITMFFAMMLLMGTLYVHMFLFARLHVKRIAALPPADGVAPQQHSCMKG
AVTITILLGVFIFCWAPFFLHLVLIITCPTNPYCICYTAHFNTYLVLIMCNSVIDPLIYA
FRSLELRNTFREILCGCNGMNLG
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| BDBM50058956 |
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| n/a |
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| Name | BDBM50058956 |
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| Synonyms: | (R)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-5-guanidino-pentanoic acid [(R)-1-carbamoyl-2-(1H-indol-3-yl)-ethyl]-amide | CHEMBL66464 |
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| Type | Small organic molecule |
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| Emp. Form. | C28H36N8O4 |
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| Mol. Mass. | 548.6366 |
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| SMILES | CC(=O)N[C@H](Cc1ccccc1)C(=O)N[C@H](CCCNC(N)=N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(N)=O |
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| Structure | 
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