| Reaction Details |
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 | Report a problem with these data |
| Target | Glucagon receptor |
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| Ligand | BDBM50059352 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_73016 (CHEMBL681695) |
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| IC50 | 19±n/a nM |
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| Citation |  Azizeh, BY; Ahn, JM; Caspari, R; Shenderovich, MD; Trivedi, D; Hruby, VJ The role of phenylalanine at position 6 in glucagon's mechanism of biological action: multiple replacement analogues of glucagon. J Med Chem40:2555-62 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Glucagon receptor |
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| Name: | Glucagon receptor |
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| Synonyms: | GL-R | GLR_RAT | Gcgr |
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| Type: | PROTEIN |
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| Mol. Mass.: | 55053.40 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_1450588 |
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| Residue: | 485 |
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| Sequence: | MLLTQLHCPYLLLLLVVLSCLPKAPSAQVMDFLFEKWKLYSDQCHHNLSLLPPPTELVCN
RTFDKYSCWPDTPPNTTANISCPWYLPWYHKVQHRLVFKRCGPDGQWVRGPRGQSWRDAS
QCQMDDDEIEVQKGVAKMYSSYQVMYTVGYSLSLGALLLALVILLGLRKLHCTRNYIHGN
LFASFVLKAGSVLVIDWLLKTRYSQKIGDDLSVSVWLSDGAVAGCRVATVIMQYGIIANY
CWLLVEGVYLYSLLSITTFSEKSFFSLYLCIGWGSPLLFVIPWVVVKCLFENVQCWTSND
NMGFWWILRIPVLLAILINFFIFVRIIHLLVAKLRAHQMHYADYKFRLARSTLTLIPLLG
VHEVVFAFVTDEHAQGTLRSTKLFFDLFFSSFQGLLVAVLYCFLNKEVQAELLRRWRRWQ
EGKALQEERMASSHGSHMAPAGTCHGDPCEKLQLMSAGSSSGTGCEPSAKTSLASSLPRL
ADSPT
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| BDBM50059352 |
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| n/a |
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| Name | BDBM50059352 |
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| Synonyms: | CHEMBL442499 | [des-His1, Trp6, Glu9] glucagon-NH2 |
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| Type | Small organic molecule |
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| Emp. Form. | C150H222N42O47S |
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| Mol. Mass. | 3397.686 |
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| SMILES | n/a |
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| Structure | 
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