| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 1 |
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| Ligand | BDBM50454937 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_200359 (CHEMBL807426) |
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| Ki | 5382±n/a nM |
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| Citation |  Yang, L; Guo, L; Pasternak, A; Mosley, R; Rohrer, S; Birzin, E; Foor, F; Cheng, K; Schaeffer, J; Patchett, AA Spiro[1H-indene-1,4'-piperidine] derivatives as potent and selective non-peptide human somatostatin receptor subtype 2 (sst2) agonists. J Med Chem41:2175-9 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 1 |
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| Name: | Somatostatin receptor type 1 |
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| Synonyms: | SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1) |
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| Type: | Enzyme |
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| Mol. Mass.: | 42692.81 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P30872 |
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| Residue: | 391 |
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| Sequence: | MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCTSRITTL
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| BDBM50454937 |
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| n/a |
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| Name | BDBM50454937 |
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| Synonyms: | CHEMBL2112223 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H37N5O2 |
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| Mol. Mass. | 499.6471 |
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| SMILES | NCCCCCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)N1CCC2(CC1)C=Cc1ccccc21 |c:32| |
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| Structure | 
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