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TargetDiamine acetyltransferase 1
LigandBDBM50095444
Substrate/Competitorn/a
Meas. Tech.ChEMBL_198446 (CHEMBL872601)
Ki 50000±n/a nM
Citation Casero, RAWoster, PM Terminally alkylated polyamine analogues as chemotherapeutic agents. J Med Chem44:1-26 (2001) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Diamine acetyltransferase 1
Name:Diamine acetyltransferase 1
Synonyms:SAT | SAT1 | SAT1_HUMAN | Spermidine/spermine N(1)-acetyltransferase 1
Type:PROTEIN
Mol. Mass.:20017.22
Organism:Homo sapiens (Human)
Description:ChEMBL_1337637
Residue:171
Sequence:
MAKFVIRPATAADCSDILRLIKELAKYEYMEEQVILTEKDLLEDGFGEHPFYHCLVAEVP
KEHWTPEGHSIVGFAMYYFTYDPWIGKLLYLEDFFVMSDYRGFGIGSEILKNLSQVAMRC
RCSSMHFLVAEWNEPSINFYKRRGASDLSSEEGWRLFKIDKEYLLKMATEE
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  Blast E-value cutoff:
BDBM50095444
n/a
NameBDBM50095444
Synonyms:CHEMBL315330 | Methyl-phosphonic acid mono-{3-[3-(3-ethylamino-propylamino)-propylamino]-propyl} ester
TypeSmall organic molecule
Emp. Form.C12H30N3O3P
Mol. Mass.295.3587
SMILESCCNCCCNCCCNCCCOP(C)(O)=O
Structure
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