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TargetMelanocortin receptor 5
LigandBDBM50144877
Substrate/Competitorn/a
Meas. Tech.ChEMBL_106668 (CHEMBL884505)
EC50 0.56±n/a nM
Citation Wilczynski, AWang, XSJoseph, CGXiang, ZBauzo, RMScott, JWSorensen, NBShaw, AMMillard, WJRichards, NGHaskell-Luevano, C Identification of putative agouti-related protein(87-132)-melanocortin-4 receptor interactions by homology molecular modeling and validation using chimeric peptide ligands. J Med Chem47:2194-207 (2004) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Melanocortin receptor 5
Name:Melanocortin receptor 5
Synonyms:MC5R_MOUSE | Mc5r | Melanocortin receptor 5 | Melanocortin receptor 5 (MC5R)
Type:Enzyme
Mol. Mass.:36966.58
Organism:Mus musculus (Mouse)
Description:P41149
Residue:325
Sequence:
MNSSSTLTVLNLTLNASEDGILGSNVKNKSLACEEMGIAVEVFLTLGLVSLLENILVIGA
IVKNKNLHSPMYFFVGSLAVADMLVSMSNAWETVTIYLLNNKHLVIADTFVRHIDNVFDS
MICISVVASMCSLLAIAVDRYITIFYALRYHHIMTARRSGVIIACIWTFCISCGIVFIIY
YESKYVIICLISMFFTMLFFMVSLYIHMFLLARNHVKRIAASPRYNSVRQRTSMKGAITL
TMLLGIFIVCWSPFFLHLILMISCPQNVYCSCFMSYFNMYLILIMCNSVIDPLIYALRSQ
EMRRTFKEIVCCHGFRRPCRLLGGY
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  Blast E-value cutoff:
BDBM50144877
n/a
NameBDBM50144877
Synonyms:CHEMBL269274
TypeSmall organic molecule
Emp. Form.C176H251N55O48S16
Mol. Mass.4418.256
SMILESn/a
Structure
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