| Reaction Details |
|---|
 | Report a problem with these data |
| Target | P2Y purinoceptor 1 |
|---|
| Ligand | BDBM50410192 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_310399 (CHEMBL833177) |
|---|
| EC50 | 9.4±n/a nM |
|---|
| Citation |  Major, DT; Nahum, V; Wang, Y; Reiser, G; Fischer, B Molecular recognition in purinergic receptors. 2. Diastereoselectivity of the h-P2Y1-receptor. J Med Chem47:4405-16 (2004) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| P2Y purinoceptor 1 |
|---|
| Name: | P2Y purinoceptor 1 |
|---|
| Synonyms: | ATP receptor | P2RY1_RAT | P2Y1 | P2ry1 | Purinergic receptor | Purinergic receptor P2Y1 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 42338.46 |
|---|
| Organism: | Rattus norvegicus |
|---|
| Description: | ChEMBL_873671 |
|---|
| Residue: | 373 |
|---|
| Sequence: | MTEVPWSAVPNGTDAAFLAGLGSLWGNSTIASTAAVSSSFRCALIKTGFQFYYLPAVYIL
VFIIGFLGNSVAIWMFVFHMKPWSGISVYMFNLALADFLYVLTLPALIFYYFNKTDWIFG
DVMCKLQRFIFHVNLYGSILFLTCISAHRYSGVVYPLKSLGRLKKKNAIYVSVLVWLIVV
VAISPILFYSGTGIRKNKTVTCYDSTSDEYLRSYFIYSMCTTVAMFCIPLVLILGCYGLI
VRALIYKDLDNSPLRRKSIYLVIIVLTVFAVSYIPFHVMKTMNLRARLDFQTPEMCDFND
RVYATYQVTRGLASLNSCVDPILYFLAGDTFRRRLSRATRKASRRSEANLQSKSEEMTLN
ILSEFKQNGDTSL
|
|
|
|---|
| BDBM50410192 |
|---|
| n/a |
|---|
| Name | BDBM50410192 |
|---|
| Synonyms: | CHEMBL2093074 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C10H16N5O12P3S |
|---|
| Mol. Mass. | 523.247 |
|---|
| SMILES | Nc1ncnc2n(cnc12)C1O[C@H](CO[P@](O)(=S)OP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1O |r| |
|---|
| Structure | 
|
|---|
Search and Browse
