| Reaction Details |
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 | Report a problem with these data |
| Target | P2Y purinoceptor 6 |
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| Ligand | BDBM50306711 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_611870 (CHEMBL1070825) |
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| EC50 | 140±n/a nM |
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| Citation |  Ginsburg-Shmuel, T; Haas, M; Schumann, M; Reiser, G; Kalid, O; Stern, N; Fischer, B 5-OMe-UDP is a potent and selective P2Y(6)-receptor agonist. J Med Chem53:1673-85 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| P2Y purinoceptor 6 |
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| Name: | P2Y purinoceptor 6 |
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| Synonyms: | P2RY6 | P2RY6_HUMAN | P2Y purinoceptor 6 | P2Y6 | Pyrimidinergic receptor P2Y6 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36452.29 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1511151 |
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| Residue: | 328 |
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| Sequence: | MEWDNGTGQALGLPPTTCVYRENFKQLLLPPVYSAVLAAGLPLNICVITQICTSRRALTR
TAVYTLNLALADLLYACSLPLLIYNYAQGDHWPFGDFACRLVRFLFYANLHGSILFLTCI
SFQRYLGICHPLAPWHKRGGRRAAWLVCVAVWLAVTTQCLPTAIFAATGIQRNRTVCYDL
SPPALATHYMPYGMALTVIGFLLPFAALLACYCLLACRLCRQDGPAEPVAQERRGKAARM
AVVVAAAFAISFLPFHITKTAYLAVRSTPGVPCTVLEAFAAAYKGTRPFASANSVLDPIL
FYFTQKKFRRRPHELLQKLTAKWQRQGR
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| BDBM50306711 |
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| n/a |
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| Name | BDBM50306711 |
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| Synonyms: | CHEMBL590441 | INS-48823 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H32N4O23P4 |
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| Mol. Mass. | 892.4403 |
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| SMILES | O[C@@H]1[C@@H](COP(O)(=O)OP(O)(=O)OP(O)(=O)OP(O)(=O)OC[C@H]2O[C@H](C3OC(Cc4ccccc4)OC23)n2ccc(=O)[nH]c2=O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O |r| |
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| Structure | 
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