| Reaction Details |
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 | Report a problem with these data |
| Target | Pancreatic triacylglycerol lipase |
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| Ligand | BDBM50381859 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_817316 (CHEMBL2025941) |
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| Ki | 360000±n/a nM |
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| Citation |  Park, S; Yu, J An approach for differentiating isozymes. Construction of libraries containing short aromatic peptides as part of a method to design selective inhibitors against lipases. Bioorg Med Chem Lett22:3147-51 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Pancreatic triacylglycerol lipase |
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| Name: | Pancreatic triacylglycerol lipase |
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| Synonyms: | LIPP_HUMAN | PL | PNLIP | Pancreatic lipase |
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| Type: | PROTEIN |
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| Mol. Mass.: | 51157.75 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_527250 |
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| Residue: | 465 |
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| Sequence: | MLPLWTLSLLLGAVAGKEVCYERLGCFSDDSPWSGITERPLHILPWSPKDVNTRFLLYTN
ENPNNFQEVAADSSSISGSNFKTNRKTRFIIHGFIDKGEENWLANVCKNLFKVESVNCIC
VDWKGGSRTGYTQASQNIRIVGAEVAYFVEFLQSAFGYSPSNVHVIGHSLGAHAAGEAGR
RTNGTIGRITGLDPAEPCFQGTPELVRLDPSDAKFVDVIHTDGAPIVPNLGFGMSQVVGH
LDFFPNGGVEMPGCKKNILSQIVDIDGIWEGTRDFAACNHLRSYKYYTDSIVNPDGFAGF
PCASYNVFTANKCFPCPSGGCPQMGHYADRYPGKTNDVGQKFYLDTGDASNFARWRYKVS
VTLSGKKVTGHILVSLFGNKGNSKQYEIFKGTLKPDSTHSNEFDSDVDVGDLQMVKFIWY
NNVINPTLPRVGASKIIVETNVGKQFNFCSPETVREEVLLTLTPC
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| BDBM50381859 |
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| n/a |
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| Name | BDBM50381859 |
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| Synonyms: | CHEMBL2022681 |
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| Type | Small organic molecule |
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| Emp. Form. | C38H38N4O5 |
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| Mol. Mass. | 630.7321 |
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| SMILES | CCCCOc1ccc(NC(=O)CCC(=O)N[C@H](C(=O)N[C@H](C(N)=O)c2ccc3ccccc3c2)c2ccc3ccccc3c2)cc1 |r| |
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| Structure | 
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