| Reaction Details |
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 | Report a problem with these data |
| Target | Kappa-type opioid receptor |
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| Ligand | BDBM50386976 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_827540 (CHEMBL2051481) |
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| Ki | >10000±n/a nM |
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| Citation |  Stavitskaya, L; Shim, J; Healy, JR; Matsumoto, RR; MacKerell, AD; Coop, A Deconstructing 14-phenylpropyloxymetopon: minimal requirements for binding to mu opioid receptors. Bioorg Med Chem20:4556-63 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Kappa-type opioid receptor |
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| Name: | Kappa-type opioid receptor |
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| Synonyms: | KOR-1 | Kappa Opioid Receptor | OPIATE Kappa | OPRK_RAT | Opioid receptor | Oprk1 | Ror-d |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 42692.90 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | P34975 |
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| Residue: | 380 |
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| Sequence: | MESPIQIFRGEPGPTCAPSACLLPNSSSWFPNWAESDSNGSVGSEDQQLEPAHISPAIPV
IITAVYSVVFVVGLVGNSLVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFQSAVYL
MNSWPFGDVLCKIVISIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKIINI
CIWLLASSVGISAIVLGGTKVREDVDVIECSLQFPDDEYSWWDLFMKICVFVFAFVIPVL
IIIVCYTLMILRLKSVRLLSGSREKDRNLRRITKLVLVVVAVFIICWTPIHIFILVEALG
STSHSTAVLSSYYFCIALGYTNSSLNPVLYAFLDENFKRCFRDFCFPIKMRMERQSTNRV
RNTVQDPASMRDVGGMNKPV
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| BDBM50386976 |
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| n/a |
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| Name | BDBM50386976 |
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| Synonyms: | CHEMBL2048971 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H27NO |
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| Mol. Mass. | 309.4452 |
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| SMILES | CN(CCCc1ccccc1)CCOC\C=C\c1ccccc1 |
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| Structure | 
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