| Reaction Details |
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 | Report a problem with these data |
| Target | Solute carrier family 2, facilitated glucose transporter member 1 |
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| Ligand | BDBM50388391 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_829819 (CHEMBL2061377) |
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| IC50 | 5000±n/a nM |
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| Citation |  Wang, D; Chu, PC; Yang, CN; Yan, R; Chuang, YC; Kulp, SK; Chen, CS Development of a novel class of glucose transporter inhibitors. J Med Chem55:3827-36 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Solute carrier family 2, facilitated glucose transporter member 1 |
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| Name: | Solute carrier family 2, facilitated glucose transporter member 1 |
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| Synonyms: | GLUT-1 | GLUT1 | GTR1_HUMAN | Glucose Transporter 1 (hGLUT1) | Glucose transporter | Glucose transporter type 1, erythrocyte/brain | HepG2 glucose transporter | SLC2A1 |
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| Type: | Protein |
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| Mol. Mass.: | 54091.71 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 492 |
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| Sequence: | MEPSSKKLTGRLMLAVGGAVLGSLQFGYNTGVINAPQKVIEEFYNQTWVHRYGESILPTT
LTTLWSLSVAIFSVGGMIGSFSVGLFVNRFGRRNSMLMMNLLAFVSAVLMGFSKLGKSFE
MLILGRFIIGVYCGLTTGFVPMYVGEVSPTALRGALGTLHQLGIVVGILIAQVFGLDSIM
GNKDLWPLLLSIIFIPALLQCIVLPFCPESPRFLLINRNEENRAKSVLKKLRGTADVTHD
LQEMKEESRQMMREKKVTILELFRSPAYRQPILIAVVLQLSQQLSGINAVFYYSTSIFEK
AGVQQPVYATIGSGIVNTAFTVVSLFVVERAGRRTLHLIGLAGMAGCAILMTIALALLEQ
LPWMSYLSIVAIFGFVAFFEVGPGPIPWFIVAELFSQGPRPAAIAVAGFSNWTSNFIVGM
CFQYVEQLCGPYVFIIFTVLLVLFFIFTYFKVPETKGRTFDEIASGFRQGGASQSDKTPE
ELFHPLGADSQV
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| BDBM50388391 |
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| n/a |
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| Name | BDBM50388391 |
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| Synonyms: | CHEMBL2057965 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H18F3NO3S |
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| Mol. Mass. | 373.39 |
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| SMILES | CCC(CC)CN1C(=O)S\C(=C/c2ccc(O)c(c2)C(F)(F)F)C1=O |
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| Structure | 
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