| Reaction Details |
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 | Report a problem with these data |
| Target | Casein kinase I isoform alpha |
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| Ligand | BDBM50215926 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_853878 (CHEMBL2154998) |
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| IC50 | 50000±n/a nM |
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| Citation |  Shengule, SR; Loa-Kum-Cheung, WL; Parish, CR; Blairvacq, M; Meijer, L; Nakao, Y; Karuso, P A one-pot synthesis and biological activity of ageladine A and analogues. J Med Chem54:2492-503 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Casein kinase I isoform alpha |
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| Name: | Casein kinase I isoform alpha |
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| Synonyms: | CK1 | CKI-alpha | CSNK1A1 | KC1A_PIG |
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| Type: | PROTEIN |
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| Mol. Mass.: | 14639.55 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_939731 |
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| Residue: | 125 |
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| Sequence: | GEEVAVKLESQKARHPQLLYESKLYKILQGGVGIPHIRWYGQEKDYNVLVMDLLGPSLED
LFNFCSRRFTMKTVLMLADQMISRIEYVHTKNFIHRDIKPDNFLMGIGRHCNKLFLIDFG
LAKKY
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| BDBM50215926 |
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| n/a |
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| Name | BDBM50215926 |
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| Synonyms: | 4-(4,5-dibromo-1H-pyrrol-2-yl)-1H-imidazo[4,5-c]pyridin-2-amine | Ageladine A | CHEMBL230806 |
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| Type | Small organic molecule |
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| Emp. Form. | C10H7Br2N5 |
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| Mol. Mass. | 357.004 |
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| SMILES | Nc1nc2c(nccc2[nH]1)-c1cc(Br)c(Br)[nH]1 |
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| Structure | 
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