| Reaction Details |
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 | Report a problem with these data |
| Target | D(3) dopamine receptor |
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| Ligand | BDBM50002310 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_877403 (CHEMBL2182833) |
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| Ki | 22±n/a nM |
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| Citation |  Spetea, M; Berzetei-Gurske, IP; Guerrieri, E; Schmidhammer, H Discovery and pharmacological evaluation of a diphenethylamine derivative (HS665), a highly potent and selective¿ opioid receptor agonist. J Med Chem55:10302-6 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(3) dopamine receptor |
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| Name: | D(3) dopamine receptor |
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| Synonyms: | DOPAMINE D3 | DRD3 | DRD3_HUMAN | Dopamine D3 receptor | Dopamine D3 receptor (D3) | Dopamine D3 receptor (D3R) | Dopamine receptor | Dopamine receptor (D3) | Dopamine receptor D3 |
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| Type: | n/a |
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| Mol. Mass.: | 44243.43 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 400 |
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| Sequence: | MASLSQLSSHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERAL
QTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILN
LCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTV
CSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQ
QTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRK
LSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHV
SPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
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| BDBM50002310 |
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| n/a |
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| Name | BDBM50002310 |
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| Synonyms: | 3-[2-(Phenethyl-propyl-amino)-ethyl]-phenol; hydrobromide | CHEMBL1188090 | CHEMBL545783 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H25NO |
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| Mol. Mass. | 283.4079 |
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| SMILES | CCCN(CCc1ccccc1)CCc1cccc(O)c1 |
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| Structure | 
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