| Reaction Details |
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 | Report a problem with these data |
| Target | Urotensin-2 receptor |
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| Ligand | BDBM50413016 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_496756 (CHEMBL1005393) |
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| Ki | 1000±n/a nM |
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| Citation |  Wang, Y; Wu, Z; Guida, BF; Lawrence, SK; Neeb, MJ; Rivero, RA; Douglas, SA; Jin, J N-alkyl-5H-pyrido[4,3-b]indol-1-amines and derivatives as novel urotensin-II receptor antagonists. Bioorg Med Chem Lett18:4936-9 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Urotensin-2 receptor |
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| Name: | Urotensin-2 receptor |
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| Synonyms: | Urotensin II receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 41170.15 |
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| Organism: | Felis catus |
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| Description: | ChEMBL_496756 |
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| Residue: | 374 |
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| Sequence: | MALSPAPLSGFPEPSAAPNASLNRSWASPTEPSSLEDLVATGAIGAVLSAMGVVGVAGNA
YTLVVMCRVLHTSASMSVYVVNLALADLLYLLSIPFIVATYVTKEWHFGDVGCRVLFSLD
FLTMHASIFTLTVMSSERYAAVLRPLDTVQRSKGYRKVLALGTWLLALLLALPMMLAIRL
VHRGHKSLCLPVWGPRAHRAYLTLLFGTSIVGPGTVIGLLYVRLARAYWLSQRASFTQTR
RLPNPKVLYLILGIVLLFWACFLPFWLWQLLAQYRGAQTLTPRTARIVNYLTTCLTYGNS
CVNPFLYTLLTKNYREYRRRSLRARSARGPAGARHSLPCRVRFQRGSGHSLCSSSQQATE
TITLSPAASRAVCA
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| BDBM50413016 |
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| n/a |
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| Name | BDBM50413016 |
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| Synonyms: | CHEMBL496516 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H13N3S |
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| Mol. Mass. | 279.36 |
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| SMILES | C(Nc1nccc2[nH]c3ccccc3c12)c1cccs1 |
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| Structure | 
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