| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide FF receptor 1 |
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| Ligand | BDBM50414852 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_590511 (CHEMBL1058558) |
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| EC50 | 79.43±n/a nM |
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| Citation |  Gaubert, G; Bertozzi, F; Kelly, NM; Pawlas, J; Scully, AL; Nash, NR; Gardell, LR; Lameh, J; Olsson, R Discovery of selective nonpeptidergic neuropeptide FF2 receptor agonists. J Med Chem52:6511-4 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Neuropeptide FF receptor 1 |
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| Name: | Neuropeptide FF receptor 1 |
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| Synonyms: | G-protein coupled receptor 147 | GPR147 | NPFF1 | NPFF1_HUMAN | NPFFR1 | RFamide-related peptide receptor OT7T022 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 47840.07 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1474637 |
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| Residue: | 430 |
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| Sequence: | MEGEPSQPPNSSWPLSQNGTNTEATPATNLTFSSYYQHTSPVAAMFIVAYALIFLLCMVG
NTLVCFIVLKNRHMHTVTNMFILNLAVSDLLVGIFCMPTTLVDNLITGWPFDNATCKMSG
LVQGMSVSASVFTLVAIAVERFRCIVHPFREKLTLRKALVTIAVIWALALLIMCPSAVTL
TVTREEHHFMVDARNRSYPLYSCWEAWPEKGMRRVYTTVLFSHIYLAPLALIVVMYARIA
RKLCQAPGPAPGGEEAADPRASRRRARVVHMLVMVALFFTLSWLPLWALLLLIDYGQLSA
PQLHLVTVYAFPFAHWLAFFNSSANPIIYGYFNENFRRGFQAAFRARLCPRPSGSHKEAY
SERPGGLLHRRVFVVVRPSDSGLPSESGPSSGAPRPGRLPLRNGRVAHHGLPREGPGCSH
LPLTIPAWDI
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| BDBM50414852 |
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| n/a |
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| Name | BDBM50414852 |
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| Synonyms: | CHEMBL573738 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H14N4O |
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| Mol. Mass. | 242.2765 |
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| SMILES | [#6]-c1ccccc1-c1ccc(-[#6]=[#7]\[#7]=[#6](\[#7])-[#7])o1 |w:11.11| |
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| Structure | 
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