Ki Summary

Reaction Details

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Target

Solute carrier organic anion transporter family member 2A1

Ligand

BDBM21544

Substrate/Competitor

n/a

Meas. Tech.

ChEMBL_836787 (CHEMBL2075312)

98±n/a nM

Citation

Pucci, ML; Bao, Y; Chan, B; Itoh, S; Lu, R; Copeland, NG; Gilbert, DJ; Jenkins, NA; Schuster, VL Cloning of mouse prostaglandin transporter PGT cDNA: species-specific substrate affinities. Am J Physiol277:734-41 (1999) [PubMed] Article

More Info.:

Get all data from this article, Assay Method

Solute carrier organic anion transporter family member 2A1

Name:

Solute carrier organic anion transporter family member 2A1

Synonyms:

Oatp2a1 | SO2A1_MOUSE | Slc21a2 | Slco2a1 | Solute carrier family 21 member 2

Type:

PROTEIN

Mol. Mass.:

70168.17

Organism:

Mus musculus

Description:

ChEMBL_836787

Residue:

643

Sequence:

MGLLPKPGARQGSGTSSVPARRCSRSVFNNIKVFVLCHGLLQLCQLLYSAYFKSSLTTIE
KRFGLSSSSSGLISSLNEISNAILIIFVSYFGSRVNRPRMIGIGGLLLAAGAFVLTLPHF
LSEPYQYASTTAGNSSHFQTDLCQKHLPGLLPSKCHSTVPDTQKETSSMWSLMVVAQLLA
GVGTVPIQPFGISYVDDFAEPTNSPLYISILFAIAVFGPAFGYLLGSVMLRIFVDYGRVD
TATVNLSPGDPRWIGAWWLGLLISSGFLIVTSLPFFFFPRAMSRGAERSVIAEETMKMEE
DKSRGSLMDFIKRFPRIFLRLLMNPLFMLVVLSQCTFSSVIAGLSTFLNKFLEKQYDASA
AYANLLIGAVNLPAAALGMLFGGILMKRFVFPLQTIPRVAATIMTISIILCAPLFFMGCS
TPAVAEVYPPSTPSSIHPQPPACRRDCLCPDSVFHPVCGDNGVEYLSPCHAGCSSLNVSS
AASKQPIYLNCSCVTGGSASAKTGSCPTSCAQLLLPSIFLISFVALIACVSHNPLYMMVL
RVVNQDEKSFAIGVQFLLMRLLAWLPSPSLYGLLIDSSCIRWNYLCSGRRGACAYYDNDA
LRNRYLGLQVIYKVLGTLLLFFISWRVKKNREYSLQENASGLI

BDBM21544

n/a

Name

BDBM21544

Synonyms:

(5Z)-7-[(1R,2R,5S)-5-hydroxy-2-[(1E,3S)-3-hydroxyoct-1-en-1-yl]-3-oxocyclopentyl]hept-5-enoic acid | 11-Dehydroprostaglandin F2 alpha | Prostaglandin D2 | [3H]PGD2

Type

radiolabeled ligand

Emp. Form.

C20H32O5

Mol. Mass.

352.4651

SMILES

CCCCC[C@H](O)\C=C\[C@@H]1[C@@H](C\C=C/CCCC(O)=O)[C@@H](O)CC1=O |r|

Structure