| Reaction Details |
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 | Report a problem with these data |
| Target | Beta-2 adrenergic receptor |
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| Ligand | BDBM50241366 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_37826 (CHEMBL653458) |
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| Kd | 44±n/a nM |
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| Citation |  IJzerman, AP; Aué, GH; Bultsma, T; Linschoten, MR; Timmerman, H Quantitative evaluation of the beta 2-adrenoceptor affinity of phenoxypropanolamines and phenylethanolamines. J Med Chem28:1328-34 (1985) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Beta-2 adrenergic receptor |
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| Name: | Beta-2 adrenergic receptor |
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| Synonyms: | ADRB2 | ADRB2_BOVIN | Beta-2 adrenergic receptor | Beta-2 adrenoceptor | Beta-2 adrenoreceptor | adrenergic Beta |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 47141.18 |
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| Organism: | BOVINE |
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| Description: | adrenergic Beta ADRB2 BOVINE::Q28044 |
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| Residue: | 418 |
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| Sequence: | MGQPGNRSVFLLAPNASHAPDQNVTLERDEAWVVGMGILMSLIVLAIVFGNVLVITAIAK
FERLQTVTNYFITSLACADLVMGLAVVPFGACHILMKMWTFGNFWCEFWTSIDVLCVTAS
IETLCVIAVDRYLAITSPFKYQCLLTKNKARVVILMVWIVSGLTSFLPIQMHWYRASHKE
AINCYAKETCCDFFTNQPYAIASSIVSFYLPLVVMVFVYSRVFQVAKRQLQKIDKSEGRF
HAQNVSQVEQDGRSGLGQRRTSKFYLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIKD
NLIRKEIYILLNWLGYINSAFNPLIYCRSPDFRIAFQELLCLRRSSLKAYGNGCSSNSND
RTDYTGEQSGYHLGEEKDSELLCEDPPGTENFVNQQGTVPSDSIDSQGRNCSTNDSLL
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| BDBM50241366 |
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| n/a |
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| Name | BDBM50241366 |
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| Synonyms: | (S)-1-(isopropylamino)-3-(m-tolyloxy)propan-2-ol | (S)-1-(isopropylamino)-3-(m-tolyloxy)propan-2-ol ((2S)-toliprolol) | CHEMBL252319 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H21NO2 |
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| Mol. Mass. | 223.3113 |
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| SMILES | CC(C)NC[C@H](O)COc1cccc(C)c1 |r| |
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| Structure | 
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