| Reaction Details |
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 | Report a problem with these data |
| Target | Platelet-activating factor receptor |
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| Ligand | BDBM50422599 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_307258 (CHEMBL830837) |
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| IC50 | 1259±n/a nM |
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| Citation |  Goldring, WP; Alexander, SP; Kendall, DA; Pattenden, G Novel phomactin analogues as PAF receptor ligands. Bioorg Med Chem Lett15:3263-6 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Platelet-activating factor receptor |
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| Name: | Platelet-activating factor receptor |
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| Synonyms: | PAF Platelet activating factor | PAF-R | PAFR | PTAFR | PTAFR_HUMAN | Platelet activating factor receptor | Platelet-activating factor receptor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 39219.60 |
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| Organism: | Homo sapiens (Human) |
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| Description: | PAF Platelet activating factor PTAFR HUMAN::P25105 |
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| Residue: | 342 |
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| Sequence: | MEPHDSSHMDSEFRYTLFPIVYSIIFVLGVIANGYVLWVFARLYPCKKFNEIKIFMVNLT
MADMLFLITLPLWIVYYQNQGNWILPKFLCNVAGCLFFINTYCSVAFLGVITYNRFQAVT
RPIKTAQANTRKRGISLSLVIWVAIVGAASYFLILDSTNTVPDSAGSGNVTRCFEHYEKG
SVPVLIIHIFIVFSFFLVFLIILFCNLVIIRTLLMQPVQQQRNAEVKRRALWMVCTVLAV
FIICFVPHHVVQLPWTLAELGFQDSKFHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLTEKFYSMRSSRKCSRATTDTVTEVVVPFNQIPGNSLKN
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| BDBM50422599 |
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| n/a |
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| Name | BDBM50422599 |
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| Synonyms: | CHEMBL372012 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H30O4 |
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| Mol. Mass. | 334.4498 |
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| SMILES | C[C@@H]1C[C@H]2O[C@@]3(C)CC\C=C(C)\CC[C@@]1(C)C1=C2[C@](O)(OC1)[C@H]3O |c:9,17| |
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| Structure | 
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