| Reaction Details |
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 | Report a problem with these data |
| Target | Scm-like with four MBT domains protein 1 |
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| Ligand | BDBM50440582 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_983406 (CHEMBL2429076) |
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| IC50 | >10000±n/a nM |
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| Citation |  James, LI; Korboukh, VK; Krichevsky, L; Baughman, BM; Herold, JM; Norris, JL; Jin, J; Kireev, DB; Janzen, WP; Arrowsmith, CH; Frye, SV Small-molecule ligands of methyl-lysine binding proteins: optimization of selectivity for L3MBTL3. J Med Chem56:7358-71 (2013) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Scm-like with four MBT domains protein 1 |
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| Name: | Scm-like with four MBT domains protein 1 |
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| Synonyms: | RU1 | Renal ubiquitous protein 1 | SFMBT1 | SMBT1_HUMAN | hSFMBT |
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| Type: | PROTEIN |
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| Mol. Mass.: | 98135.34 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_104121 |
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| Residue: | 866 |
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| Sequence: | MNGEQQLDADAGSGMEEVELSWEDYLEETGSTAVPYGSFKHVDTRLQNGFAPGMKLEVAV
RTDPETYWVATVITTCEQLLLLRYDGYGEDRRADFWCDIRKADLYPIGWCEQNKKTLEAP
EGIRDKVSDWDEFLRQTLIGACSPPVPLLEGLRNGRNPLDLIAPGSRLECQAFQDSLSTW
IVTVVENIGGRLKLRYEGLESSDNYEHWLYYLDPFLHHVGWAAQQGYELQPPSAIRHLKN
EAEWQEILAKVKEEEEEPLPSYLFKDKQVIGIHTFSVNMKLEAVDPWSPFGISPATVVKV
FDEKYFLVEMDDLRPENHARRSFVCHADSPGIFPVQWSLKNGLHISPPPGYPSQDFDWAD
YLKQCGAEAAPQRCFPPLISEHEFKENMKLEAVNPILPEEVCVATITAVRGSYLWLQLEG
SKKPIPECIVSVESMDIFPLGWCETNGHPLSTPRRARVYKQRKIAVVQPEKQVPSSRTVH
EGLRNQELNSTESVMINGKYCCPKIYFNHRCFSGPYLNKGRIAELPQCVGPGNCVLVLRE
VLTLLINAAYKPSRVLRELQLDKDSVWHGCGEVLKAKYKGKSYRATVEIVKTADRVTEFC
RQTCIKLECCPNLFGPRMVLDKCSENCSVLTKTKYTHYYGKKKNKRIGRPPGGHSNLACA
LKKASKRRKRRKNVFVHKKKRSSASVDNTPAGSPQGSGGEDEDDPDEGDDDSLSEGSTSE
QQDELQEESEMSEKKSCSSSPTQSEISTSLPPDRQRRKRELRTFSFSDDENKPPSPKEIR
IEVAERLHLDSNPLKWSVADVVRFIRSTDCAPLARIFLDQEIDGQALLLLTLPTVQECMD
LKLGPAIKLCHHIERIKFAFYEQFAN
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| BDBM50440582 |
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| n/a |
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| Name | BDBM50440582 |
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| Synonyms: | CHEMBL2426463 |
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| Type | Small organic molecule |
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| Emp. Form. | C24H36N4O2 |
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| Mol. Mass. | 412.5682 |
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| SMILES | O=C(NCCCN1CCCC1)c1ccc(cc1)C(=O)N1CCC(CC1)N1CCCC1 |
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| Structure | 
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