| Reaction Details |
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 | Report a problem with these data |
| Target | Acrosin |
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| Ligand | BDBM50010106 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1344334 (CHEMBL3257004) |
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| Ki | 680±n/a nM |
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| Citation |  Parrish, RF; Straus, JW; Paulson, JD; Polakoski, KL; Tidwell, RR; Geratz, JD; Stevens, FM Structure-activity relationships for the inhibition of acrosin by benzamidine derivatives. J Med Chem21:1132-6 (1979) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Acrosin |
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| Name: | Acrosin |
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| Synonyms: | 53 kDa fucose-binding protein | ACR | ACRO_PIG | Acrosin heavy chain | Acrosin light chain |
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| Type: | PROTEIN |
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| Mol. Mass.: | 45383.66 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_108297 |
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| Residue: | 415 |
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| Sequence: | MLPTAVLLVLAVSVAARDNATCDGPCGLRFRQKLESGMRVVGGMSAEPGAWPWMVSLQIF
MYHNNRRYHTCGGILLNSHWVLTAAHCFKNKKKVTDWRLIFGANEVVWGSNKPVKPPLQE
RFVEEIIIHEKYVSGLEINDIALIKITPPVPCGPFIGPGCLPQFKAGPPRAPQTCWVTGW
GYLKEKGPRTSPTLQEARVALIDLELCNSTRWYNGRIRSTNVCAGYPRGKIDTCQGDSGG
PLMCRDRAENTFVVVGITSWGVGCARAKRPGVYTSTWPYLNWIASKIGSNALQMVQLGTP
PRPSTPAPPVRPPSVQTPVRPPWYFQRPPGPSQQPGSRPRPPAPPPAPPPPPPPPPPPPP
PPPPPPQQVSAKPPQALSFAKRLQQLIEALKGTAFSSGRSYYETETTDLQELPAS
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| BDBM50010106 |
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| n/a |
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| Name | BDBM50010106 |
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| Synonyms: | CHEMBL2418012 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H15BrN4O |
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| Mol. Mass. | 347.21 |
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| SMILES | NC(=N)c1ccc(COc2ccc(cc2Br)C(N)=N)cc1 |
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| Structure | 
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