| Reaction Details |
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 | Report a problem with these data |
| Target | Uracil nucleotide/cysteinyl leukotriene receptor |
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| Ligand | BDBM50010475 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1353474 (CHEMBL3269457) |
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| Ki | 1630±n/a nM |
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| Citation |  Köse, M; Ritter, K; Thiemke, K; Gillard, M; Kostenis, E; Müller, CE Development of [(3)H]2-Carboxy-4,6-dichloro-1H-indole-3-propionic Acid ([(3)H]PSB-12150): A Useful Tool for Studying GPR17. ACS Med Chem Lett5:326-30 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Uracil nucleotide/cysteinyl leukotriene receptor |
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| Name: | Uracil nucleotide/cysteinyl leukotriene receptor |
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| Synonyms: | GPR17 | GPR17_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 41013.71 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1353471 |
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| Residue: | 367 |
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| Sequence: | MSKRSWWAGSRKPPREMLKLSGSDSSQSMNGLEVAPPGLITNFSLATAEQCGQETPLENM
LFASFYLLDFILALVGNTLALWLFIRDHKSGTPANVFLMHLAVADLSCVLVLPTRLVYHF
SGNHWPFGEIACRLTGFLFYLNMYASIYFLTCISADRFLAIVHPVKSLKLRRPLYAHLAC
AFLWVVVAVAMAPLLVSPQTVQTNHTVVCLQLYREKASHHALVSLAVAFTFPFITTVTCY
LLIIRSLRQGLRVEKRLKTKAVRMIAIVLAIFLVCFVPYHVNRSVYVLHYRSHGASCATQ
RILALANRITSCLTSLNGALDPIMYFFVAEKFRHALCNLLCGKRLKGPPPSFEGKTNESS
LSAKSEL
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| BDBM50010475 |
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| n/a |
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| Name | BDBM50010475 |
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| Synonyms: | GAVESTINEL | GV-150526X |
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| Type | Small organic molecule |
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| Emp. Form. | C18H12Cl2N2O3 |
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| Mol. Mass. | 375.205 |
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| SMILES | OC(=O)c1[nH]c2cc(Cl)cc(Cl)c2c1\C=C\C(=O)Nc1ccccc1 |
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| Structure | 
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