| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50010483 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1353487 (CHEMBL3269823) |
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| IC50 | 1.4±n/a nM |
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| Citation |  Ballet, S; Betti, C; Novoa, A; Tömböly, C; Nielsen, CU; Helms, HC; Lesniak, A; Kleczkowska, P; Chung, NN; Lipkowski, AW; Brodin, B; Tourwé, D; Schiller, PW In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt ACS Med Chem Lett5:352-357 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
|
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|
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| BDBM50010483 |
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| n/a |
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| Name | BDBM50010483 |
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| Synonyms: | CHEMBL2181202 |
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| Type | Small organic molecule |
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| Emp. Form. | C32H49N9O5 |
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| Mol. Mass. | 639.7888 |
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| SMILES | Cc1cc(O)cc(C)c1C[C@H](N)C(=O)N[C@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCCN)C(N)=O |r| |
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| Structure | 
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