| Reaction Details |
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 | Report a problem with these data |
| Target | Oxoeicosanoid receptor 1 |
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| Ligand | BDBM50046281 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1447591 (CHEMBL3373786) |
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| IC50 | 460±n/a nM |
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| Citation |  Gore, V; Chourey, S; Ye, Q; Patel, P; Ouedraogo, Y; Gravel, S; Powell, WS; Rokach, J Base-dependent formation of cis and trans olefins and their application in the synthesis of 5-oxo-ETE receptor antagonists. Bioorg Med Chem Lett24:3385-8 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Oxoeicosanoid receptor 1 |
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| Name: | Oxoeicosanoid receptor 1 |
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| Synonyms: | 5-oxo-ETE G-protein coupled receptor | G-protein coupled receptor 170 | G-protein coupled receptor R527 | G-protein coupled receptor TG1019 | GPR170 | OXER1 | OXER1_HUMAN | Oxoeicosanoid receptor 1 | TG 1019 | TG1019 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 45833.20 |
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| Organism: | Homo sapiens (Human) |
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| Description: | TG 1019 0 HUMAN::Q8TDS5 |
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| Residue: | 423 |
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| Sequence: | MLCHRGGQLIVPIIPLCPEHSCRGRRLQNLLSGPWPKQPMELHNLSSPSPSLSSSVLPPS
FSPSPSSAPSAFTTVGGSSGGPCHPTSSSLVSAFLAPILALEFVLGLVGNSLALFIFCIH
TRPWTSNTVFLVSLVAADFLLISNLPLRVDYYLLHETWRFGAAACKVNLFMLSTNRTASV
VFLTAIALNRYLKVVQPHHVLSRASVGAAARVAGGLWVGILLLNGHLLLSTFSGPSCLSY
RVGTKPSASLRWHQALYLLEFFLPLALILFAIVSIGLTIRNRGLGGQAGPQRAMRVLAMV
VAVYTICFLPSIIFGMASMVAFWLSACRSLDLCTQLFHGSLAFTYLNSVLDPVLYCFSSP
NFLHQSRALLGLTRGRQGPVSDESSYQPSRQWRYREASRKAEAIGKLKVQGEVSLEKEGS
SQG
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| BDBM50046281 |
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| n/a |
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| Name | BDBM50046281 |
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| Synonyms: | CHEMBL3311230 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H24ClNO3 |
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| Mol. Mass. | 361.862 |
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| SMILES | CCCC\C=C/c1cc2ccc(Cl)cc2n1C(=O)CC(C)CC(O)=O |
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| Structure | 
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