| Reaction Details |
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 | Report a problem with these data |
| Target | Serine racemase |
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| Ligand | BDBM50055465 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1450503 (CHEMBL3380621) |
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| IC50 | 520000±n/a nM |
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| Citation |  Mori, H; Wada, R; Li, J; Ishimoto, T; Mizuguchi, M; Obita, T; Gouda, H; Hirono, S; Toyooka, N In silico and pharmacological screenings identify novel serine racemase inhibitors. Bioorg Med Chem Lett24:3732-5 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Serine racemase |
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| Name: | Serine racemase |
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| Synonyms: | SRR | SRR_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36565.80 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1516972 |
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| Residue: | 340 |
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| Sequence: | MCAQYCISFADVEKAHINIRDSIHLTPVLTSSILNQLTGRNLFFKCELFQKTGSFKIRGA
LNAVRSLVPDALERKPKAVVTHSSGNHGQALTYAAKLEGIPAYIVVPQTAPDCKKLAIQA
YGASIVYCEPSDESRENVAKRVTEETEGIMVHPNQEPAVIAGQGTIALEVLNQVPLVDAL
VVPVGGGGMLAGIAITVKALKPSVKVYAAEPSNADDCYQSKLKGKLMPNLYPPETIADGV
KSSIGLNTWPIIRDLVDDIFTVTEDEIKCATQLVWERMKLLIEPTAGVGVAAVLSQHFQT
VSPEVKNICIVLSGGNVDLTSSITWVKQAERPASYQSVSV
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| BDBM50055465 |
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| n/a |
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| Name | BDBM50055465 |
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| Synonyms: | CHEMBL3317754 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H14BrFN2O3 |
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| Mol. Mass. | 381.196 |
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| SMILES | Fc1ccc(OCC(=O)NCC(=O)Nc2ccc(Br)cc2)cc1 |
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| Structure | 
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