| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50078763 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1472324 (CHEMBL3419674) |
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| Ki | 2.8±n/a nM |
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| Citation |  Ogawa, G; Tius, MA; Zhou, H; Nikas, SP; Halikhedkar, A; Mallipeddi, S; Makriyannis, A 3'-functionalized adamantyl cannabinoid receptor probes. J Med Chem58:3104-16 (2015) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CNR2_MOUSE | Cannabinoid CB2 receptor | Cannabinoid receptor | Cannabinoid receptor 2 | Cnr2 | mCB2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38220.43 |
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| Organism: | MOUSE |
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| Description: | P47936 |
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| Residue: | 347 |
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| Sequence: | MEGCRETEVTNGSNGGLEFNPMKEYMILSSGQQIAVAVLCTLMGLLSALENMAVLYIILS
SRRLRRKPSYLFISSLAGADFLASVIFACNFVIFHVFHGVDSNAIFLLKIGSVTMTFTAS
VGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALCVMWVLSALISYLPLMGWTCCPSPCS
ELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHRHVATLAEHQDRQVPGIARMRLD
VRLAKTLGLVLAVLLICWFPALALMGHSLVTTLSDQVKEAFAFCSMLCLVNSMVNPIIYA
LRSGEIRSAAQHCLIGWKKYLQGLGPEGKEEGPRSSVTETEADVKTT
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| BDBM50078763 |
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| n/a |
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| Name | BDBM50078763 |
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| Synonyms: | CHEMBL3416122 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H33NO3 |
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| Mol. Mass. | 407.5451 |
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| SMILES | [H][C@@]12C[C@H](O)CC[C@@]1([H])C(C)(C)Oc1cc(cc(O)c21)[C@@]12CC3CC(C[C@](C3)(C1)C#N)C2 |r,TLB:23:24:21.22.27:28,27:22:31:26.28.25,27:26:31:21.22.23| |
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| Structure | 
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