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TargetSomatostatin receptor type 4
LigandBDBM50155308
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1565560
Ki 1170±n/a nM
Citation FridÚn-Saxin MSeifert TMalo Mda Silva Andersson KPemberton NDyrager CFriberg ADahlÚn KWallÚn EAGr°tli MLuthman K Chroman-4-one and chromone based somatostatin▀-turn mimetics. Eur J Med Chem 114:59-64 (2016) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Somatostatin receptor type 4
Name:Somatostatin receptor type 4
Synonyms:SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SST4R | Somatostatin receptor type 4 (SSTR4)
Type:Enzyme
Mol. Mass.:42015.38
Organism:Homo sapiens (Human)
Description:P31391
Residue:388
Sequence:
MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLV
GLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCR
AVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLP
IAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRA
VALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILS
YANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCM
CPPLPCQQEALQPEPGRKRIPLTRTTTF
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  Blast E-value cutoff:
BDBM50155308
n/a
NameBDBM50155308
Synonyms:CHEMBL3780791
TypeSmall organic molecule
Emp. Form.C24H24Cl3NO2
Mol. Mass.464.812
SMILESCl.Cl.NCCCc1cc(Cl)cc2c1oc(CCc1cccc3ccccc13)cc2=O
Structure
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