| Reaction Details |
|---|
 | Report a problem with these data |
| Target | RYamide receptor |
|---|
| Ligand | BDBM50192747 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_1613599 (CHEMBL3855399) |
|---|
| EC50 | 5900±n/a nM |
|---|
| Citation |  Yoon, YK; Kim, JH; Kim, JH; Kwon, JY; Kim, YC; Kim, YJ; Park, ZY Pyrazolodiazepine derivatives with agonist activity toward Drosophila RYamide receptor. Bioorg Med Chem Lett26:5116-5118 (2016) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| RYamide receptor |
|---|
| Name: | RYamide receptor |
|---|
| Synonyms: | NPY-R | NepYr | Neuropeptide Y-like receptor | RYAR_DROME | RYa-R | RYamide receptor | Synonyms=NepYr |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 53538.04 |
|---|
| Organism: | Drosophila melanogaster |
|---|
| Description: | ChEMBL_116973 |
|---|
| Residue: | 464 |
|---|
| Sequence: | MEHHNSHLLPGGSEKMYYIAHQQPMLRNEDDNYQEGYFIRPDPASLIYNTTALPADDEGS
NYGYGSTTTLSGLQFETYNITVMMNFSCDDYDLLSEDMWSSAYFKIIVYMLYIPIFIFAL
IGNGTVCYIVYSTPRMRTVTNYFIASLAIGDILMSFFCVPSSFISLFILNYWPFGLALCH
FVNYSQAVSVLVSAYTLVAISIDRYIAIMWPLKPRITKRYATFIIAGVWFIALATALPIP
IVSGLDIPMSPWHTKCEKYICREMWPSRTQEYYYTLSLFALQFVVPLGVLIFTYARITIR
VWAKRPPGEAETNRDQRMARSKRKMVKMMLTVVIVFTCCWLPFNILQLLLNDEEFAHWDP
LPYVWFAFHWLAMSHCCYNPIIYCYMNARFRSGFVQLMHRMPGLRRWCCLRSVGDRMNAT
SGTGPALPLNRMNTSTTYISARRKPRATSLRANPLSCGETSPLR
|
|
|
|---|
| BDBM50192747 |
|---|
| n/a |
|---|
| Name | BDBM50192747 |
|---|
| Synonyms: | CHEMBL3935892 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C31H42N6O4 |
|---|
| Mol. Mass. | 562.703 |
|---|
| SMILES | Cc1noc(C)c1CN1CC(Cc2ccccc2)NC(=O)c2nn(CCC3CCN(CC3)C(=O)OC(C)(C)C)cc12 |
|---|
| Structure | 
|
|---|
Search and Browse
