Reaction Details |
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Target | Fatty acid-binding protein 5 |
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Ligand | BDBM50197087 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_1619187 (CHEMBL3861356) |
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Ki | 100±n/a nM |
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Citation | Kühne, H; Obst-Sander, U; Kuhn, B; Conte, A; Ceccarelli, SM; Neidhart, W; Rudolph, MG; Ottaviani, G; Gasser, R; So, SS; Li, S; Zhang, X; Gao, L; Myers, M Design and synthesis of selective, dual fatty acid binding protein 4 and 5 inhibitors. Bioorg Med Chem Lett26:5092-5097 (2016) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Fatty acid-binding protein 5 |
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Name: | Fatty acid-binding protein 5 |
Synonyms: | FABP5 | FABP5_HUMAN | Fatty acid binding protein epidermal | Fatty acid-binding protein 5 (FABP5) |
Type: | Enzyme |
Mol. Mass.: | 15164.79 |
Organism: | Homo sapiens (Human) |
Description: | Q01469 |
Residue: | 135 |
Sequence: | MATVQQLEGRWRLVDSKGFDEYMKELGVGIALRKMGAMAKPDCIITCDGKNLTIKTESTL
KTTQFSCTLGEKFEETTADGRKTQTVCNFTDGALVQHQEWDGKESTITRKLKDGKLVVEC
VMNNVTCTRIYEKVE
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BDBM50197087 |
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n/a |
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Name | BDBM50197087 |
Synonyms: | CHEMBL3950316 |
Type | Small organic molecule |
Emp. Form. | C22H21ClN2O2 |
Mol. Mass. | 380.867 |
SMILES | Cc1cc(Cl)cc2c(-c3ccccc3)c(C(O)=O)c(nc12)N1CCCCC1 |
Structure |
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