Reaction Details |
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Target | Somatostatin receptor type 3 |
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Ligand | BDBM82256 |
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Substrate/Competitor | n/a |
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Ki | 177±n/a nM |
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Comments | PDSP_385 |
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Citation | Shimon, I; Taylor, JE; Dong, JZ; Bitonte, RA; Kim, S; Morgan, B; Coy, DH; Culler, MD; Melmed, S Somatostatin receptor subtype specificity in human fetal pituitary cultures. Differential role of SSTR2 and SSTR5 for growth hormone, thyroid-stimulating hormone, and prolactin regulation. J Clin Invest99:789-98 (1997) [PubMed] Article |
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More Info.: | Get all data from this article |
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Somatostatin receptor type 3 |
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Name: | Somatostatin receptor type 3 |
Synonyms: | SOMATOSTATIN SST3 | SS-3-R | SS3-R | SS3R | SSR-28 | SSR3_HUMAN | SSTR3 | Somatostatin receptor type 3 (SSTR3) |
Type: | Protein |
Mol. Mass.: | 45855.97 |
Organism: | Homo sapiens (Human) |
Description: | P32745 |
Residue: | 418 |
Sequence: | MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLL
GNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVM
AVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVV
FSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRV
WAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVA
LPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEE
SREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL
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BDBM82256 |
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n/a |
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Name | BDBM82256 |
Synonyms: | BIM 23056 | CAS_150155-61-6 | D-Phe-Phe-Tyr-D-Trp-Lys-Val-Phe-D-Nal-NH2 | DC-25-20 |
Type | Small organic molecule |
Emp. Form. | C71H81N11O9 |
Mol. Mass. | 1232.4711 |
SMILES | CC(C)[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](N)Cc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](Cc1ccc2ccccc2c1)C(N)=O |r| |
Structure |
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