Reaction Details |
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Target | Somatostatin receptor type 3 |
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Ligand | BDBM85052 |
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Substrate/Competitor | n/a |
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Ki | 26.8±n/a nM |
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Comments | PDSP_3373 |
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Citation | Shimon, I; Taylor, JE; Dong, JZ; Bitonte, RA; Kim, S; Morgan, B; Coy, DH; Culler, MD; Melmed, S Somatostatin receptor subtype specificity in human fetal pituitary cultures. Differential role of SSTR2 and SSTR5 for growth hormone, thyroid-stimulating hormone, and prolactin regulation. J Clin Invest99:789-98 (1997) [PubMed] Article |
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More Info.: | Get all data from this article |
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Somatostatin receptor type 3 |
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Name: | Somatostatin receptor type 3 |
Synonyms: | SOMATOSTATIN SST3 | SS-3-R | SS3-R | SS3R | SSR-28 | SSR3_HUMAN | SSTR3 | Somatostatin receptor type 3 (SSTR3) |
Type: | Protein |
Mol. Mass.: | 45855.97 |
Organism: | Homo sapiens (Human) |
Description: | P32745 |
Residue: | 418 |
Sequence: | MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLL
GNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVM
AVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVV
FSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRV
WAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVA
LPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEE
SREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL
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BDBM85052 |
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n/a |
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Name | BDBM85052 |
Synonyms: | BIM 23197 | BIM-23197 |
Type | Small organic molecule |
Emp. Form. | C57H81N13O13S3 |
Mol. Mass. | 1252.527 |
SMILES | n/a |
Structure |
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