| Reaction Details |
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 | Report a problem with these data |
| Target | Gamma-aminobutyric acid receptor subunit rho-3 |
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| Ligand | BDBM23183 |
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| Substrate/Competitor | n/a |
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| Ki | 460±n/a nM |
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| Comments | PDSP_1260 |
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| Citation |  Chang, Y; Covey, DF; Weiss, DS Correlation of the apparent affinities and efficacies of gamma-aminobutyric acid(C) receptor agonists. Mol Pharmacol58:1375-80 (2000) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Gamma-aminobutyric acid receptor subunit rho-3 |
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| Name: | Gamma-aminobutyric acid receptor subunit rho-3 |
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| Synonyms: | GABA B rho 1 | GABRR3 | GBRR3_HUMAN | Gamma-aminobutyric acid receptor subunit rho-3 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 54281.08 |
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| Organism: | Homo sapiens (Human) |
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| Description: | GABA B rho 1 0 HUMAN::A8MPY1 |
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| Residue: | 467 |
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| Sequence: | MVLAFQLVSFTYIWIILKPNVCAASNIKMTHQRCSSSMKQTCKQETRMKKDDSTKARPQK
YEQLLHIEDNDFAMRPGFGGSPVPVGIDVHVESIDSISETNMDFTMTFYLRHYWKDERLS
FPSTANKSMTFDHRLTRKIWVPDIFFVHSKRSFIHDTTMENIMLRVHPDGNVLLSLRITV
SAMCFMDFSRFPLDTQNCSLELESYAYNEDDLMLYWKHGNKSLNTEEHMSLSQFFIEDFS
ASSGLAFYSSTGWYNRLFINFVLRRHVFFFVLQTYFPAILMVMLSWVSFWIDRRAVPARV
SLGITTVLTMSTIITAVSASMPQVSYLKAVDVYLWVSSLFVFLSVIEYAAVNYLTTVEER
KQFKKTGKISRMYNIDAVQAMAFDGCYHDSEIDMDQTSLSLNSEDFMRRKSICSPSTDSS
RIKRRKSLGGHVGRIILENNHVIDTYSRILFPIVYILFNLFYWGVYV
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| BDBM23183 |
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| n/a |
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| Name | BDBM23183 |
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| Synonyms: | 5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL273481 | Muscimol | Pantherine |
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| Type | GABA Agonist |
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| Emp. Form. | C4H6N2O2 |
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| Mol. Mass. | 114.1026 |
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| SMILES | NCc1cc(=O)[nH]o1 |
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| Structure | 
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