| Reaction Details |
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 | Report a problem with these data |
| Target | Solute carrier organic anion transporter family member 2A1 |
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| Ligand | BDBM85719 |
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| Substrate/Competitor | n/a |
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| Ki | 5000±n/a nM |
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| Comments | PDSP_1466 |
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| Citation |  Schuster, VL; Itoh, S; Andrews, SW; Burk, RM; Chen, J; Kedzie, KM; Gil, DW; Woodward, DF Synthetic modification of prostaglandin f(2alpha) indicates different structural determinants for binding to the prostaglandin F receptor versus the prostaglandin transporter. Mol Pharmacol58:1511-6 (2000) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Solute carrier organic anion transporter family member 2A1 |
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| Name: | Solute carrier organic anion transporter family member 2A1 |
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| Synonyms: | OATP2A1 | Prostaglandin Transporter | SLC21A2 | SLCO2A1 | SO2A1_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 70068.67 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Prostaglandin Transporter 0 HUMAN::Q92959 |
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| Residue: | 643 |
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| Sequence: | MGLLPKLGASQGSDTSTSRAGRCARSVFGNIKVFVLCQGLLQLCQLLYSAYFKSSLTTIE
KRFGLSSSSSGLISSLNEISNAILIIFVSYFGSRVHRPRLIGIGGLFLAAGAFILTLPHF
LSEPYQYTLASTGNNSRLQAELCQKHWQDLPPSKCHSTTQNPQKETSSMWGLMVVAQLLA
GIGTVPIQPFGISYVDDFSEPSNSPLYISILFAISVFGPAFGYLLGSVMLQIFVDYGRVN
TAAVNLVPGDPRWIGAWWLGLLISSALLVLTSFPFFFFPRAMPIGAKRAPATADEARKLE
EAKSRGSLVDFIKRFPCIFLRLLMNSLFVLVVLAQCTFSSVIAGLSTFLNKFLEKQYGTS
AAYANFLIGAVNLPAAALGMLFGGILMKRFVFSLQAIPRIATTIITISMILCVPLFFMGC
STPTVAEVYPPSTSSSIHPQSPACRRDCSCPDSIFHPVCGDNGIEYLSPCHAGCSNINMS
SATSKQLIYLNCSCVTGGSASAKTGSCPVPCAHFLLPAIFLISFVSLIACISHNPLYMMV
LRVVNQEEKSFAIGVQFLLMRLLAWLPSPALYGLTIDHSCIRWNSLCLGRRGACAYYDND
ALRDRYLGLQMGYKALGMLLLCFISWRVKKNKEYNVQKAAGLI
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| BDBM85719 |
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| n/a |
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| Name | BDBM85719 |
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| Synonyms: | PGF2 Alpha, 1-isopropyl ester |
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| Type | Small organic molecule |
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| Emp. Form. | C23H40O5 |
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| Mol. Mass. | 396.5607 |
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| SMILES | CCCCCC(O)C=CC1C(O)CC(O)C1CC=CCCCC(=O)OC(C)C |w:7.6,17.17| |
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| Structure | 
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