| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM85734 |
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| Substrate/Competitor | n/a |
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| Ki | 0.222±n/a nM |
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| Comments | PDSP_3258 |
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| Citation |  Schiller, PW; Nguyen, TM; Berezowska, I; Dupuis, S; Weltrowska, G; Chung, NN; Lemieux, C Synthesis and in vitro opioid activity profiles of DALDA analogues. Eur J Med Chem35:895-901 (2000) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM85734 |
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| n/a |
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| Name | BDBM85734 |
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| Synonyms: | H-Hmt-D-Arg-Phe-Lys-NH2 I | H-Hmt-D-Arg-Phe-Lys-NH2 II | H-Mmt-D-Arg-Phe-Lys-NH2 |
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| Type | Small organic molecule |
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| Emp. Form. | C31H47N9O5 |
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| Mol. Mass. | 625.7622 |
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| SMILES | [#6]-c1cc(-[#8])ccc1-[#6]-[#6@H](-[#7])-[#6](=O)-[#7]-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccccc1)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6](-[#7])=O |
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| Structure | 
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