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TargetNorepinephrine transporter
LigandBDBM85092
Substrate/Competitorn/a
Ki>10000±n/a nM
CommentsPDSP_1504
Citation Millan, MJCussac, DMilligan, GCarr, CAudinot, VGobert, ALejeune, FRivet, JMBrocco, MDuqueyroix, DNicolas, JPBoutin, JANewman-Tancredi, A Antiparkinsonian agent piribedil displays antagonist properties at native, rat, and cloned, human alpha(2)-adrenoceptors: cellular and functional characterization. J Pharmacol Exp Ther297:876-87 (2001) [PubMed]
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Norepinephrine transporter
Name:Norepinephrine transporter
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:2082.45
Organism:RAT
Description:Norepinephrine transporter 0 RAT::Q9JIA2
Residue:19
Sequence:
MLLARMKPQVQPELGGADQ
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BDBM85092
n/a
NameBDBM85092
Synonyms:CAS_3605-01-4 | NSC_4850 | Piribedil
TypeSmall organic molecule
Emp. Form.C16H18N4O2
Mol. Mass.298.3397
SMILESC(N1CCN(CC1)c1ncccn1)c1ccc2OCOc2c1
Structure
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