| Reaction Details |
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 | Report a problem with these data |
| Target | Retinoic acid receptor RXR-alpha |
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| Ligand | BDBM86153 |
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| Substrate/Competitor | n/a |
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| Ki | 7600±n/a nM |
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| Comments | PDSP_3006 |
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| Citation |  Patel, S; Krause, SM; Hamill, T; Chaudhary, A; Burns, DH; Gibson, RA In vitro characterization of [3H]MethoxyPyEP, an mGluR5 selective radioligand. Life Sci73:371-9 (2003) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Retinoic acid receptor RXR-alpha |
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| Name: | Retinoic acid receptor RXR-alpha |
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| Synonyms: | NR2B Channel Blocker | Nr2b1 | RXRA_RAT | Retinoic acid receptor RXR-alpha | Retinoid X receptor alpha | Rxra |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 51273.78 |
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| Organism: | RAT |
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| Description: | NR2B Channel Blocker 0 RAT::Q05343 |
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| Residue: | 467 |
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| Sequence: | MDTKHFLPLDFSTQVNSSSLSSPTGRGSMAAPSLHPSLGPGLGSPLGSPGQLHSPISTLS
SPINGMGPPFSVISSPMGPHSMSVPTTPTLGFETGSPQLNSPMNPVSSSEDIKPPLGLNG
VLKVPAHPSGNMSSFTKHICAICGDRSSGKHYGVYSCEGCKGFFKRTVRKDLTYTCRDNK
DCLIDKRQRNRCQYCRYQKCLAMGMKREAVQEERQRGKDRNENEVESTSSANEDMPVEKI
LEAELAVEPKTETYVEANMGLNPSSPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLD
DQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVS
KMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRF
AKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQTT
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| BDBM86153 |
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| n/a |
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| Name | BDBM86153 |
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| Synonyms: | CAS_180081 | MK-801 | NSC_180081 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H15N |
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| Mol. Mass. | 221.297 |
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| SMILES | CC12NC(Cc3ccccc13)c1ccccc21 |TLB:9:10:2:11.16,6:5:2:11.16,THB:12:11:10.5.4:2,15:16:10.5.4:2| |
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| Structure | 
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