| Reaction Details |
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 | Report a problem with these data |
| Target | Cyclin-dependent kinase 2 |
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| Ligand | BDBM7163 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Thermofluor |
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| pH | 7.5±n/a |
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| Temperature | 298.15±n/a K |
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| Kd | 4960±n/a nM |
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| Citation |  CSARdock, CD CDK2 in CSAR_FULL_RELEASE_3JULY2012 CSAR1:0 (2012) |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Cyclin-dependent kinase 2 |
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| Name: | Cyclin-dependent kinase 2 |
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| Synonyms: | CDK2 | CDK2-Kinase | CDK2_HUMAN | CDKN2 | Cell division protein kinase 2 | Cyclin-dependent kinase 2 (CDK2) | Protein cereblon/Cyclin-dependent kinase 2 | p33 protein kinase |
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| Type: | Enzyme Subunit |
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| Mol. Mass.: | 33938.17 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P24941 |
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| Residue: | 298 |
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| Sequence: | MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNH
PNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHS
HRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYY
STAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSF
PKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL
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| BDBM7163 |
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| n/a |
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| Name | BDBM7163 |
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| Synonyms: | 3-Phenylacetamidoaminopyrazole deriv. 40 | CS10 | N-(5-Cyclopropyl-1H-pyrazol-3-yl)-2-(4-thien-2-ylphenyl)acetamide | N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-[4-(thiophen-2-yl)phenyl]acetamide |
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| Type | Small organic molecule |
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| Emp. Form. | C18H17N3OS |
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| Mol. Mass. | 323.412 |
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| SMILES | O=C(Cc1ccc(cc1)-c1cccs1)Nc1cc(n[nH]1)C1CC1 |
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| Structure | 
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