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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Neuropeptide Y receptor type 5 | ||
| Ligand | BDBM118181 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Binding Assay | ||
| pH | 7.4±n/a | ||
| Temperature | 298.15±n/a K | ||
| IC50 | 1.8±n/a nM | ||
| Comments | extracted | ||
| Citation |  Yoshida, H; Tonogaki, K; Sakagami, M; Takaya, K Cyclohexane derivative having NPY Y5 receptor antagonism US Patent US8653125 Publication Date 2/18/2014 | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Neuropeptide Y receptor type 5 | |||
| Name: | Neuropeptide Y receptor type 5 | ||
| Synonyms: | NPY-Y5 | NPY5R_MOUSE | Neuropeptide Y receptor Y5 | Neuropeptide Y receptor type 5 (NPY Y5) | Npy5 | Npy5r | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 52807.91 | ||
| Organism: | Mus musculus (Mouse) | ||
| Description: | O70342 | ||
| Residue: | 466 | ||
| Sequence: |
| ||
| BDBM118181 | |||
| n/a | |||
| Name | BDBM118181 | ||
| Synonyms: | US8653125, Ia-43 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C20H19F3N4O2 | ||
| Mol. Mass. | 404.3857 | ||
| SMILES | FC(F)(F)c1cccc(c1)-c1c[nH]c(n1)[C@@H]1CC[C@@H](CC1)NC(=O)c1ccon1 |r,wU:18.23,15.16,(9.7,-.62,;8.37,-1.39,;9.14,-2.73,;7.6,-.06,;7.04,-2.16,;7.04,-3.7,;5.7,-4.47,;4.37,-3.7,;4.37,-2.16,;5.7,-1.39,;3.04,-1.39,;3.04,.15,;1.57,.62,;.67,-.62,;1.57,-1.87,;-.67,.15,;-.67,1.69,;-2,2.46,;-3.33,1.69,;-3.33,.15,;-2,-.62,;-4.67,2.46,;-6,1.69,;-6,.15,;-7.34,2.46,;-8.8,1.98,;-9.7,3.23,;-8.8,4.47,;-7.34,4,)| | ||
| Structure | 
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