| Reaction Details |
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 | Report a problem with these data |
| Target | Prostaglandin E2 receptor EP1 subtype |
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| Ligand | BDBM119457 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Cell Response Assay |
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| IC50 | 35±n/a nM |
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| Citation |  Tatani, K; Kawamura, N; Kondo, T; Kondo, A Indole derivative or pharmaceutically acceptable salt thereof US Patent US8680120 Publication Date 3/25/2014 |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostaglandin E2 receptor EP1 subtype |
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| Name: | Prostaglandin E2 receptor EP1 subtype |
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| Synonyms: | PE2R1_RAT | Prostanoid EP1 receptor | Ptger1 |
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| Type: | Enzyme |
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| Mol. Mass.: | 43080.10 |
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| Organism: | Rattus norvegicus (Rat) |
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| Description: | P70597 |
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| Residue: | 405 |
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| Sequence: | MSPYGLNLSLVDEATTCVTPRVPNTSVVLPTGGNGTSPALPIFSMTLGAVSNVLALALLA
QVAGRLRRRRSTATFLLFVASLLAIDLAGHVIPGALVLRLYTAGRAPAGGACHFLGGCMV
FFGLCPLLLGCGMAVERCVGVTQPLIHAARVSVARARLALALLAAMALAVALLPLVHVGH
YELQYPGTWCFISLGPPGGWRQALLAGLFAGLGLAALLAALVCNTLSGLALLRARWRRRR
SRRFRENAGPDDRRRWGSRGLRLASASSASSITSTTAALRSSRGGGSARRVHAHDVEMVG
QLVGIMVVSCICWSPLLVLVVLAIGGWNSNSLQRPLFLAVRLASWNQILDPWVYILLRQA
MLRQLLRLLPLRVSAKGGPTELSLTKSAWEASSLRSSRHSGFSHL
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| BDBM119457 |
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| n/a |
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| Name | BDBM119457 |
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| Synonyms: | US8680120, 9-25 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H17NO3S |
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| Mol. Mass. | 363.43 |
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| SMILES | COc1ccc2n(Cc3cccc(c3)C(O)=O)c(cc2c1)-c1ccsc1 |
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| Structure | 
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